含多種成分:假荊芥酸(nepetalic acid),假荊芥內酯(nepetalactone),β-丁香烯(β-caryophyllene),假荊芥酐(nepetaic anhydride),9-表假荊芥內酯(9-epinepetalactone),二氫假荊芥內酯(dihydronepetalactone),異二氫假荊芥內酯(isodihydronepetalactone),假荊芥酮酸甲酯(methyl nepetonate),異假荊芥內酯(isonepetalactone), 丁香油酚(eugenol),5,9-去氫假荊芥內酯(5,9-dehydronepetalactone),4αS,7S,7αR-假荊芥酰胺(4αS,7S,7αR-2-nepetalactam),4αS,7S,7αR-2-(3R,4R,4αR,7S,7αR-八氫-4,7-二甲基-1-氧代環戊烷[C]吡喃-3-基)假荊芥酰胺[4αS,7S,7αR-2-(3R,4R,4αR,7S,7αR-octahydro-4,7-dimethyl-1-oxocyclopenta[C]pyran-3-yl)nepetalactam]和假荊茶酸甙(nepetariaside)。
葉含咖啡酰丙醇二酸(caffeoyltartronic acid),假荊芥內酯甙(nepetaside), 獼猴桃堿(actinidine),1,5,9-表去氧馬錢子甙酸(1,5,9-epideoxyloganic acid)。